Potent and selective disruption of protein kinase D functionality by a benzoxoloazepinolone

Medicine & Life Sciences

• CID755673 100%
• protein kinase D 72%
• Phorbol Esters 16%
• polo-like kinase 1 11%
• High-Throughput Screening Assays 10%
• Small Molecule Libraries 10%
• Fluorescence Polarization 10%
• Vesicular Stomatitis 9%
• Diglycerides 9%
• Histone Deacetylases 8%
• Protein-Serine-Threonine Kinases 8%
• Enzymes 8%
• Second Messenger Systems 8%
• National Institutes of Health (U.S.) 7%
• Pathologic Processes 7%
• Glycoproteins 6%
• Cell Movement 6%
• Protein Isoforms 6%
• Prostatic Neoplasms 6%
• Adenosine Triphosphate 5%
• Phosphotransferases 5%
• Cell Membrane 5%
• Animal Models 5%
• Viruses 5%
• Pharmacology 5%
• Cell Proliferation 5%

Chemical Compounds

• Phorbol 31%
• Protein 18%
• Enzyme Inhibition 13%
• Threonine 12%
• Histone 12%
• High Throughput Screening 12%
• Serine 10%
• Glycoprotein 10%
• Fragmentation 9%
• Enzyme Activity 9%
• Polarization 8%
• Molecule 7%
• Plasma 7%
• Fluorescence 6%